Compile Data Set for Download or QSAR
Found 55 of ic50 data for polymerid = 50004854
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381135(CHEMBL2017736)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381134(CHEMBL2017735)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381136(CHEMBL2017737)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381139(CHEMBL2017871)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381131(CHEMBL2017732)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381129(CHEMBL2017730)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381132(CHEMBL2017733)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381133(CHEMBL2017734)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381124(CHEMBL2017725)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381130(CHEMBL2017731)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381123(CHEMBL2017724)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381120(CHEMBL2017721)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381117(CHEMBL2017717)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381119(CHEMBL2017719)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381127(CHEMBL2017728)copy SMILEScopy InChI
Affinity DataIC50: 88nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381112(CHEMBL2017712)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381126(CHEMBL2017727)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381128(CHEMBL2017729)copy SMILEScopy InChI
Affinity DataIC50: 121nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381106(CHEMBL2017870)copy SMILEScopy InChI
Affinity DataIC50: 176nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381105(CHEMBL2017720)copy SMILEScopy InChI
Affinity DataIC50: 202nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381125(CHEMBL2017726)copy SMILEScopy InChI
Affinity DataIC50: 217nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381110(CHEMBL2017710)copy SMILEScopy InChI
Affinity DataIC50: 223nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381118(CHEMBL2017718)copy SMILEScopy InChI
Affinity DataIC50: 241nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381107(CHEMBL2017707)copy SMILEScopy InChI
Affinity DataIC50: 322nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381121(CHEMBL2017722)copy SMILEScopy InChI
Affinity DataIC50: 354nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381114(CHEMBL2017714)copy SMILEScopy InChI
Affinity DataIC50: 375nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381115(CHEMBL2017715)copy SMILEScopy InChI
Affinity DataIC50: 384nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381116(CHEMBL2017716)copy SMILEScopy InChI
Affinity DataIC50: 393nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381113(CHEMBL2017713)copy SMILEScopy InChI
Affinity DataIC50: 428nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381111(CHEMBL2017711)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381108(CHEMBL2017708)copy SMILEScopy InChI
Affinity DataIC50: 453nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381122(CHEMBL2017723)copy SMILEScopy InChI
Affinity DataIC50: 715nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421673(CHEMBL5283441)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381138(CHEMBL2017739)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381109(CHEMBL2017709)copy SMILEScopy InChI
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421686(CHEMBL5282194)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50293701(CHEMBL549536 | N-(5-methyl-1H-pyrazol-3-yl)-2-(pyr...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50293150(CHEMBL468963 | D3RKN_26 | GSK screening, 38 | N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421679(CHEMBL5282708)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421671(CHEMBL5266831)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50381137(CHEMBL2017738)copy SMILEScopy InChI
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z16JXPubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421672(CHEMBL5316225)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421685(CHEMBL5280226)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421687(CHEMBL5277580)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421681(CHEMBL5273566)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421683(CHEMBL5283041)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421676(CHEMBL5283475)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421680(CHEMBL5277737)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421682(CHEMBL5285809)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
MRC Technology

Curated by ChEMBL
LigandPNGBDBM50421684(CHEMBL5277619)copy SMILEScopy InChI
Affinity DataIC50: 6.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
Displayed 1 to 50 (of 55 total ) | Next | Last >>
Jump to: